Treatment-emergent AEs, n (%) | Grade 1 | Grade 2 | Grade 3 | Grade 4 | Any grade |
---|---|---|---|---|---|
Diarrhea | 14 (45.2) | 9 (29.0) | 5 (16.1) | 0 | 28 (90.3) |
Fatigue | 2 (6.5) | 11 (35.5) | 4 (12.9) | 1 (3.2) | 18 (58.1) |
Nausea | 9 (29.0) | 6 (19.4) | 1 (3.2) | 0 | 16 (51.6) |
Edema peripheral | 6 (19.4) | 5 (16.1) | 1 (3.2) | 0 | 12 (38.7) |
Vomiting | 7 (22.6) | 3 (9.7) | 1 (3.2) | 0 | 11 (35.5) |
Abdominal pain | 3 (9.7) | 3 (9.7) | 3 (9.7) | 0 | 9 (29.0) |
Insomnia | 7 (22.6) | 2 (6.5) | 0 | 0 | 9 (29.0) |
Pruritus | 4 (12.9) | 4 (12.9) | 1 (3.2) | 0 | 9 (29.0) |
Pain in extremity | 5 (16.1) | 2 (6.5) | 0 | 1 (3.2) | 8 (25.8) |
Night sweats | 4 (12.9) | 3 (9.7) | 0 | 0 | 7 (22.6) |
Anemia | 0 | 1 (3.2) | 3 (9.7) | 2 (6.5) | 6 (19.4) |
Bone pain | 1 (3.2) | 1 (3.2) | 4 (12.9) | 0 | 6 (19.4) |
Asthenia | 4 (12.9) | 1 (3.2) | 0 | 0 | 5 (16.1) |
Constipation | 5 (16.1) | 0 | 0 | 0 | 5 (16.1) |
Dyspnea | 4 (12.9) | 0 | 1 (3.2) | 0 | 5 (16.1) |
Cardiac murmur | 0 | 4 (12.9) | 0 | 0 | 4 (12.9) |
Hyperuricemia | 2 (6.5) | 0 | 0 | 2 (6.5) | 4 (12.9) |
Pyrexia | 4 (12.9) | 0 | 0 | 0 | 4 (12.9) |
Rash | 2 (6.5) | 1 (3.2) | 1 (3.2) | 0 | 4 (12.9) |
Upper respiratory tract infection | 3 (9.7) | 1 (3.2) | 0 | 0 | 4 (12.9) |
Weight decreased | 4 (12.9) | 0 | 0 | 0 | 4 (12.9) |